Benefits
Rapid onset anticoagulant effect
Prevents formation and extension of blood clots
Essential for surgical and dialysis procedures
Widely used in hospital and ICU settings
BP-compliant sterile injectable formulation
Usage Instructions
Administered intravenously (IV) or subcutaneously (SC) by healthcare professionals
Dosage based on body weight and coagulation parameters
Monitor activated partial thromboplastin time (aPTT) during therapy
Use under strict medical supervision
Mechanism of Action
Heparin enhances the activity of antithrombin III, which inactivates thrombin (Factor IIa) and Factor Xa. This prevents conversion of fibrinogen to fibrin, thereby inhibiting clot formation and extension.
Indications
Heparin Injection BP 5000 IU/5mL is indicated for:
Prevention and treatment of deep vein thrombosis (DVT)
Pulmonary embolism (PE)
Acute coronary syndromes
Prevention of clot formation during surgery
Anticoagulation during dialysis
Disseminated intravascular coagulation (DIC) management
Side Effects
Possible side effects include:
Bleeding
Thrombocytopenia
Injection site irritation
Hypersensitivity reactions
Osteoporosis (with prolonged use)
Precautions
Regular monitoring of coagulation parameters required
Use cautiously in patients with bleeding disorders
Monitor platelet counts to detect HIT
Avoid intramuscular injection
Use in pregnancy only if clearly indicated
Contraindications
Active major bleeding
Severe thrombocytopenia
History of heparin-induced thrombocytopenia (HIT)
Hypersensitivity to heparin
Severe uncontrolled hypertension